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Relationship between Tumor Biomarkers and Efficacy in EMILIA, a Phase III Study of Trastuzumab Emtansine in HER2-Positive Metastatic Breast Cancer.

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Clin Cancer Res2016PMID 26920887PMC5485412stubpubmedProvenance
Source
PubMed
Retrieved
Sep 8, 2026
Layer
normalized (units and labels harmonized; values unchanged)
Run
ING-CIVIC-20260908-000001
Published

Abstract

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Linked entities

Linked entities (16)

How each link was made (MeSH, dictionary, registry reference, curation…) and whether it has been validated. Candidate links are not counted in entity statistics.

Validated 16

Curated evidence

Evidence citing this paper (15)

civicProvenance
Source
CIViC — Clinical Interpretation of Variants in Cancer
Dataset
CIViC evidence items
Version
civic-2026-09-08
Retrieved
Sep 8, 2026
Layer
normalized (units and labels harmonized; values unchanged)
Evidence
expert curation
License
CC0 1.0
PMID
26920887
Run
ING-CIVIC-20260908-000001
Open at source
CuratedShowing 1–15 of 15 evidence items · levels, directions and significance as curated at the source; each row links to its CIViC record.
TherapyCancerTypeLevelDirection · significanceRating (1–5)StatusEvidenceSource
ERBB3 Overexpression1
Trastuzumab EmtansineHER2-Positive Breast CarcinomaALIASPredictiveBDoes Not Support Resistance2accepted
EID8707

In a phase 3 clinical trial (NCT00829166), metastatic HER-2 amplified breast cancer patients whose tumors harbored higher than median levels of ERBB3 mRNA treated with ado-trastuzumab emtansine (T-DM1… (full text at CIViC)

PMID 26920887 · Baselga et al., 2016 · Open in CIViC

civic
PIK3CA C420R2
TrastuzumabHER2-Positive Breast CarcinomaALIASPredictiveDSupports Resistance2accepted
EID8549

As part of a pre-clinical experiment, the efficacy of trastuzumab was evaluated against various HER2 positive cell lines. EFM-192A cell line expressing PIK3CA C420R was associated with resistance to t… (full text at CIViC)

PMID 26920887 · Baselga et al., 2016 · Open in CIViC

civic
Trastuzumab EmtansineHER2-Positive Breast CarcinomaALIASPredictiveDDoes Not Support Resistance3accepted
EID2346

As part of a pre-clinical experiment, the efficacy of ado-trastuzumab emtansine (T-DM1) was compared to that of trastuzumab against various HER2 positive cell lines. EFM-192A cell line expressing PIK3… (full text at CIViC)

PMID 26920887 · Baselga et al., 2016 · Open in CIViC

civic
PIK3CA E545K2
TrastuzumabHER2-Positive Breast CarcinomaALIASPredictiveDSupports Resistance2accepted
EID8547

As part of a pre-clinical experiment, the efficacy of trastuzumab was evaluated against various HER2 positive cell lines. MCF7-neo/HER2 cell line harboring PIK3CA E545K was associated with resistance … (full text at CIViC)

PMID 26920887 · Baselga et al., 2016 · Open in CIViC

civic
Trastuzumab EmtansineHER2-Positive Breast CarcinomaALIASPredictiveDDoes Not Support Resistance3accepted
EID2036

As part of a pre-clinical experiment, the efficacy of ado-trastuzumab emtansine (T-DM1) was compared to that of trastuzumab against various HER2 positive cell lines. MCF7-neo/HER2 cell line harboring … (full text at CIViC)

PMID 26920887 · Baselga et al., 2016 · Open in CIViC

civic
PIK3CA H1047R2
TrastuzumabHER2-Positive Breast CarcinomaALIASPredictiveDSupports Resistance2accepted
EID8548

As part of a pre-clinical experiment, the efficacy of trastuzumab was evaluated against various HER2 positive cell lines. CC1954 and KPL-4 cell lines expressing PIK3CA H1047R were associated with resi… (full text at CIViC)

PMID 26920887 · Baselga et al., 2016 · Open in CIViC

civic
Trastuzumab EmtansineHER2-Positive Breast CarcinomaALIASPredictiveDDoes Not Support Resistance3accepted
EID2103

As part of a pre-clinical experiment, the efficacy of ado-trastuzumab emtansine (T-DM1) was compared to that of trastuzumab against various HER2 positive cell lines. HCC1954 and KPL-4 cell lines expre… (full text at CIViC)

PMID 26920887 · Baselga et al., 2016 · Open in CIViC

civic
PIK3CA I391M2
TrastuzumabHER2-Positive Breast CarcinomaALIASPredictiveDDoes Not Support Resistance2accepted
EID8663

As part of a pre-clinical experiment, the efficacy of trastuzumab was evaluated against various HER2 positive cell lines using cell viability assays. ZR-75-30 cell line expressing PIK3CA I391M was ass… (full text at CIViC)

PMID 26920887 · Baselga et al., 2016 · Open in CIViC

civic
Trastuzumab EmtansineHER2-Positive Breast CarcinomaALIASPredictiveDDoes Not Support Resistance3accepted
EID2867

As part of a pre-clinical experiment, the efficacy of ado-trastuzumab emtansine (T-DM1) was evaluated against various HER2 positive cell lines. ZR-75-30 cell line expressing PIK3CA I391M was associate… (full text at CIViC)

PMID 26920887 · Baselga et al., 2016 · Open in CIViC

civic
PIK3CA K111N3
TrastuzumabHER2-Positive Breast CarcinomaALIASPredictiveDSupports Resistance3rejected
EID8550

As part of a pre-clinical experiment, the efficacy of trastuzumab was compared to that of ado-trastuzumab emtansine (T-DM1) against various HER2 positive cell lines. BT-474 cell line expressing PIK3CA… (full text at CIViC)

PMID 26920887 · Baselga et al., 2016 · Open in CIViC

civic
〃HER2-Positive Breast CarcinomaALIASPredictiveDDoes Not Support Resistance2accepted
EID8662

As part of a pre-clinical experiment, the efficacy of trastuzumab was evaluated against various HER2 positive cell lines in cell viability assays. BT-474 cell line expressing PIK3CA K111N was associat… (full text at CIViC)

PMID 26920887 · Baselga et al., 2016 · Open in CIViC

civic
Trastuzumab EmtansineHER2-Positive Breast CarcinomaALIASPredictiveDDoes Not Support Resistance3accepted
EID2866

As part of a pre-clinical experiment, the efficacy of ado-trastuzumab emtansine (T-DM1) was evaluated against various HER2 positive cell lines. BT-474 cell line expressing PIK3CA K111N was associated … (full text at CIViC)

PMID 26920887 · Baselga et al., 2016 · Open in CIViC

civic
PIK3CA Mutation2
Capecitabine + LapatinibCombinationHER2-Positive Breast CarcinomaALIASPredictiveBSupports Resistance3accepted
EID8705

In a phase 3 clinical trial (NCT00829166), metastatic HER-2 amplified breast cancer patients whose tumors harbored PIK3CA mutations treated with standard of care capecitabine and lapatinib combination… (full text at CIViC)

PMID 26920887 · Baselga et al., 2016 · Open in CIViC

civic
Trastuzumab EmtansineHER2-Positive Breast CarcinomaALIASPredictiveBDoes Not Support Resistance3accepted
EID8536

In a phase 3 clinical trial (NCT00829166), metastatic HER-2 amplified breast cancer patients whose tumors harbored PIK3CA mutations treated with ado-trastuzumab emtansine (T-DM1; n=40) were associated… (full text at CIViC)

PMID 26920887 · Baselga et al., 2016 · Open in CIViC

civic
PTEN Loss1
Trastuzumab EmtansineHER2-Positive Breast CarcinomaALIASPredictiveBDoes Not Support Resistance3accepted
EID8706

In a phase 3 clinical trial (NCT00829166), metastatic HER-2 amplified breast cancer patients whose tumors had decreased, slightly decreased, or absent PTEN expression (assessed by IHC) treated with ad… (full text at CIViC)

PMID 26920887 · Baselga et al., 2016 · Open in CIViC

civic