Loading drugs…
Loading drugs…
Drugs
One entity per molecule (INN preferred); brand names and development codes are aliases. Approvals are always shown with jurisdiction and indication.
819 drugs
| Drug | Kind | Mechanism | Approvals | Evidence items | Trials | Identifiers |
|---|---|---|---|---|---|---|
| Vincristine | Small Molecule | Tubulin inhibitor | 8 | 4 | 870 | C933 · CHEMBL90555 |
| Dostarlimab | Monoclonal Antibody | Programmed cell death protein 1 antagonist | 8 | 3 | 89 | C126799 · CHEMBL4298124 |
| Prednisolone | Small Molecule | Glucocorticoid receptor agonist | 8 | 3 | 129 | C769 · CHEMBL131 |
| Apalutamide | Small Molecule | Androgen Receptor antagonist | 8 | 1 | 107 | C92574 · CHEMBL3183409 |
| Carmustine | Small Molecule | Glutathione reductase inhibitor; DNA inhibitor; RNA inhibitor | 8 | 1 | 191 | C349 · CHEMBL513 |
| Epcoritamab | Monoclonal Antibody | B-lymphocyte antigen CD20 binding agent; T cell surface glycoprotein CD3 binding agent | 8 | 0 | 59 | CHEMBL4650393 |
| Ibritumomab Tiuxetan | Monoclonal Antibody | — | 8 | 0 | 28 | CHEMBL1201606 |
| Ifosfamide | Small Molecule | DNA inhibitor | 8 | 0 | 314 | CHEMBL1024 |
| Ofatumumab | Monoclonal Antibody | B-lymphocyte antigen CD20 binding agent | 8 | 0 | 82 | CHEMBL1201836 |
| Retifanlimab | Monoclonal Antibody | Programmed cell death protein 1 antagonist | 8 | 0 | 65 | CHEMBL4298037 |
| Sodium Iodide 131 I | Small Molecule | — | 8 | 0 | 1 | CHEMBL1201084 |
| Thyrotropin Alfa | Other | Thyroid stimulating hormone receptor agonist | 8 | 0 | 5 | CHEMBL1201533 |
| Triptorelin | Other | Gonadotropin-releasing hormone receptor agonist | 8 | 0 | 63 | CHEMBL1201334 |
| Lapatinib | Small Molecule | Receptor protein-tyrosine kinase erbB-2 inhibitor; Epidermal growth factor receptor erbB1 inhibitor | 7 | 86 | 222 | C26653 · CHEMBL554 |
| Alectinib | Small Molecule | ALK tyrosine kinase receptor inhibitor; Tyrosine-protein kinase receptor RET inhibitor; EML4-ALK inhibitor | 7 | 41 | 61 | C101790 · CHEMBL1738797 |
| Midostaurin | Small Molecule | Tyrosine-protein kinase receptor FLT3 inhibitor; Stem cell growth factor receptor inhibitor; Platelet-derived growth factor receptor inhibitor; Protein kinase C (PKC) inhibitor; Vascular endothelial growth factor receptor 2 inhibitor | 7 | 33 | 43 | C1872 · CHEMBL608533 |
| Cobimetinib | Small Molecule | Dual specificity mitogen-activated protein kinase kinase 1 inhibitor; Dual specificity mitogen-activated protein kinase kinase 2 inhibitor | 7 | 22 | 87 | C68923 · CHEMBL2146883 |
| Regorafenib | Small Molecule | Tyrosine-protein kinase ABL inhibitor; Serine/threonine-protein kinase RAF inhibitor; Stem cell growth factor receptor inhibitor; Fibroblast growth factor receptor 1 inhibitor; MAP kinase p38 beta inhibitor; Fibroblast growth factor receptor 2 inhibitor; Tyrosine-protein kinase FRK inhibitor; Discoidin domain-containing receptor 2 inhibitor; Serine/threonine-protein kinase B-raf inhibitor; Tyrosine-protein kinase TIE-2 inhibitor; Platelet-derived growth factor receptor inhibitor; Vascular endothelial growth factor receptor inhibitor; Tyrosine-protein kinase receptor RET inhibitor; Ephrin type-A receptor 2 inhibitor; Nerve growth factor receptor Trk-A inhibitor | 7 | 19 | 244 | C184955 · CHEMBL1946170 |
| Sotorasib | Small Molecule | GTPase KRas inhibitor | 7 | 19 | 45 | C154287 · CHEMBL4535757 |
| Temsirolimus | Small Molecule | FK506-binding protein 1A inhibitor | 7 | 16 | 175 | C1844 · CHEMBL1201182 |
| Pemigatinib | Small Molecule | Fibroblast growth factor receptor 2 inhibitor; Fibroblast growth factor receptor 3 inhibitor; Fibroblast growth factor receptor 1 inhibitor | 7 | 7 | 44 | C121553 · CHEMBL4297522 |
| Trabectedin | Small Molecule | DNA inhibitor | 7 | 6 | 74 | C1691 · CHEMBL450449 |
| Tovorafenib | Small Molecule | RAF serine/threonine protein kinase inhibitor | 7 | 2 | 14 | C106254 · CHEMBL3348923 |
| Tucatinib | Small Molecule | Receptor protein-tyrosine kinase erbB-2 inhibitor | 7 | 2 | 55 | C77896 · CHEMBL3989868 |
| Gemtuzumab Ozogamicin | Adc | Myeloid cell surface antigen CD33 binding agent; DNA disrupting agent | 7 | 1 | 89 | C1806 · CHEMBL1201506 |
| Nilutamide | Small Molecule | Androgen Receptor antagonist | 7 | 1 | 10 | C1173 · CHEMBL1274 |
| Selinexor | Small Molecule | Exportin-1 inhibitor | 7 | 1 | 153 | C102546 · CHEMBL3545185 |
| Buserelin | Other | Gonadotropin-releasing hormone receptor agonist | 7 | 0 | 6 | CHEMBL2110824 |
| Diethylstilbestrol | Small Molecule | Estrogen receptor alpha agonist | 7 | 0 | 1 | CHEMBL411 |
| Interferon Beta-1b | Other | Interferon alpha/beta receptor agonist | 7 | 0 | 3 | CHEMBL1201563 |
| Mosunetuzumab | Monoclonal Antibody | T cell surface glycoprotein CD3 binding agent; B-lymphocyte antigen CD20 binding agent | 7 | 0 | 50 | CHEMBL4297788 |
| Pegaspargase | Other | Asparagine hydrolytic enzyme | 7 | 0 | 126 | CHEMBL2108546 |
| Peginterferon Beta-1a | Other | Interferon alpha/beta receptor agonist | 7 | 0 | 0 | CHEMBL2108677 |
| Pirtobrutinib | Small Molecule | Tyrosine-protein kinase BTK inhibitor | 7 | 0 | 52 | CHEMBL4650485 |
| Plerixafor | Small Molecule | C-X-C chemokine receptor type 4 partial agonist | 7 | 0 | 82 | CHEMBL18442 |
| Teclistamab | Monoclonal Antibody | T cell surface glycoprotein CD3 binding agent; Tumor necrosis factor receptor superfamily member 17 binding agent | 7 | 0 | 57 | CHEMBL4594505 |
| Zanidatamab | Monoclonal Antibody | Receptor protein-tyrosine kinase erbB-2 inhibitor | 7 | 0 | 29 | CHEMBL4650256 |
| Capivasertib | Small Molecule | Serine/threonine-protein kinase AKT inhibitor | 6 | 42 | 55 | C102564 · CHEMBL2325741 |
| Vandetanib | Small Molecule | Tyrosine-protein kinase SRC inhibitor; Tyrosine-protein kinase BRK inhibitor; Tyrosine-protein kinase TIE-2 inhibitor; Vascular endothelial growth factor receptor inhibitor; Tyrosine-protein kinase receptor RET inhibitor; Ephrin receptor inhibitor; Epidermal growth factor receptor inhibitor | 6 | 10 | 99 | C2737 · CHEMBL24828 |
| Repotrectinib | Small Molecule | Nerve growth factor receptor Trk-A inhibitor; Neurotrophic tyrosine kinase receptor type 2 inhibitor; Proto-oncogene tyrosine-protein kinase ROS inhibitor; NT-3 growth factor receptor inhibitor; CD74-ROS1 inhibitor; ROS1-SDC4 inhibitor | 6 | 8 | 14 | C133821 · CHEMBL4298138 |
| Decitabine | Small Molecule | DNA (cytosine-5)-methyltransferase 3A inhibitor; DNA (cytosine-5)-methyltransferase 1 inhibitor; DNA inhibitor | 6 | 4 | 287 | C981 · CHEMBL1201129 |
| Dacarbazine | Small Molecule | DNA inhibitor | 6 | 1 | 156 | C411 · CHEMBL476 |
| Ixazomib | Small Molecule | 26S proteasome inhibitor | 6 | 1 | 114 | C97940 · CHEMBL2141296 |
| Bleomycin | — | DNA inhibitor | 6 | 0 | 125 | CHEMBL6067492 |
| Dactinomycin | Other | DNA inhibitor | 6 | 0 | 50 | CHEMBL1554 |
| Darolutamide | Small Molecule | Androgen Receptor antagonist | 6 | 0 | 96 | CHEMBL4297185 |
| Dasatinib (dasatinib (s)-Propylene Glycol) | — | — | 6 | 0 | 0 | — |
| Ibandronic Acid | Small Molecule | Farnesyl diphosphate synthase inhibitor | 6 | 0 | 20 | CHEMBL997 |
| Lurbinectedin | Small Molecule | DNA negative modulator | 6 | 0 | 59 | CHEMBL4297516 |
| Mitoxantrone | Small Molecule | DNA topoisomerase II alpha inhibitor; DNA inhibitor | 6 | 0 | 217 | CHEMBL58 |