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Drugs
One entity per molecule (INN preferred); brand names and development codes are aliases. Approvals are always shown with jurisdiction and indication.
819 drugs
| Drug | Kind | Mechanism | Approvals | Evidence items | Trials | Identifiers |
|---|---|---|---|---|---|---|
| Goserelin | Other | Gonadotropin-releasing hormone receptor agonist | 13 | 0 | 194 | CHEMBL1201247 |
| Hydroxyurea | Small Molecule | Ribonucleoside-diphosphate reductase RR1 inhibitor | 13 | 0 | 65 | CHEMBL467 |
| Obinutuzumab | Monoclonal Antibody | B-lymphocyte antigen CD20 binding agent | 13 | 0 | 259 | CHEMBL1743048 |
| Pazopanib | Small Molecule | Macrophage colony stimulating factor receptor inhibitor; Stem cell growth factor receptor inhibitor; Tyrosine-protein kinase LCK inhibitor; Fibroblast growth factor receptor 3 inhibitor; Fibroblast growth factor receptor 1 inhibitor; Platelet-derived growth factor receptor inhibitor; Vascular endothelial growth factor receptor inhibitor; Tyrosine-protein kinase ITK/TSK inhibitor | 12 | 27 | 208 | C74547 · CHEMBL477772 |
| Alpelisib | Small Molecule | PI3-kinase p110-alpha subunit inhibitor | 12 | 22 | 81 | C94214 · CHEMBL2396661 |
| Mitomycin | Small Molecule | DNA inhibitor | 12 | 7 | 129 | C1820 · CHEMBL105 |
| Avelumab | Monoclonal Antibody | Programmed cell death 1 ligand 1 other | 12 | 3 | 235 | C116870 · CHEMBL3833373 |
| Enfortumab Vedotin | Adc | Nectin-4 binding agent; Tubulin inhibitor | 12 | 1 | 72 | C114500 · CHEMBL3301589 |
| Eribulin | Small Molecule | Tubulin inhibitor | 12 | 1 | 167 | C96748 · CHEMBL1683590 |
| Flutamide | Small Molecule | Androgen Receptor antagonist | 12 | 1 | 52 | C509 · CHEMBL806 |
| Pomalidomide | Small Molecule | CRL4(CRBN) E3 ubiquitin ligase inhibitor | 12 | 1 | 238 | C72560 · CHEMBL43452 |
| Interferon Alpha-2a | — | — | 12 | 0 | 5 | — |
| Axitinib | Small Molecule | Vascular endothelial growth factor receptor inhibitor | 11 | 57 | 160 | C38718 · CHEMBL1289926 |
| Ribociclib | Small Molecule | Cyclin-dependent kinase 4 inhibitor; Cyclin-dependent kinase 6 inhibitor | 11 | 12 | 155 | C95701 · CHEMBL3545110 |
| Dexamethasone | Small Molecule | Glucocorticoid receptor agonist | 11 | 5 | 1,461 | C422 · CHEMBL384467 |
| Exemestane | Small Molecule | Cytochrome P450 19A1 inhibitor | 11 | 4 | 212 | C1097 · CHEMBL1200374 |
| Fludarabine | Small Molecule | — | 11 | 1 | 1,319 | C1094 · CHEMBL1568 |
| Anagrelide | Small Molecule | Phosphodiesterase 3 inhibitor | 11 | 0 | 2 | CHEMBL760 |
| Busulfan | Small Molecule | DNA inhibitor | 11 | 0 | 373 | CHEMBL820 |
| Elotuzumab | Monoclonal Antibody | SLAM family member 7 inhibitor | 11 | 0 | 63 | CHEMBL1743010 |
| Glatiramer | — | — | 11 | 0 | 1 | — |
| Gefitinib | Small Molecule | Epidermal growth factor receptor erbB1 inhibitor | 10 | 186 | 265 | C1855 · CHEMBL939 |
| Panitumumab | Monoclonal Antibody | Epidermal growth factor receptor erbB1 inhibitor | 10 | 127 | 182 | C1857 · CHEMBL1201827 |
| Selumetinib | Small Molecule | Dual specificity mitogen-activated protein kinase kinase 1 inhibitor; Dual specificity mitogen-activated protein kinase kinase 2 inhibitor | 10 | 85 | 116 | C66939 · CHEMBL1614701 |
| Larotrectinib | Small Molecule | Neurotrophic tyrosine kinase receptor inhibitor | 10 | 79 | 20 | C115977 · CHEMBL3889654 |
| Ponatinib | Small Molecule | Bcr/Abl fusion protein inhibitor | 10 | 69 | 64 | C95777 · CHEMBL1171837 |
| Rucaparib | Small Molecule | PARP 1, 2 and 3 inhibitor | 10 | 32 | 60 | C137800 · CHEMBL1173055 |
| Asciminib | Small Molecule | Tyrosine-protein kinase ABL inhibitor; Bcr/Abl fusion protein inhibitor | 10 | 4 | 27 | C114494 · CHEMBL4208229 |
| Vinorelbine | Small Molecule | Tubulin inhibitor | 10 | 4 | 319 | C1275 · CHEMBL553025 |
| Celecoxib | Small Molecule | Cyclooxygenase-2 inhibitor | 10 | 3 | 194 | C1728 · CHEMBL118 |
| Belzutifan | Small Molecule | Endothelial PAS domain-containing protein 1 inhibitor | 10 | 1 | 34 | C135627 · CHEMBL4585668 |
| Roflumilast | Small Molecule | Phosphodiesterase 4 inhibitor | 10 | 1 | 4 | C76890 · CHEMBL193240 |
| Isatuximab | Monoclonal Antibody | Lymphocyte differentiation antigen CD38 inhibitor | 10 | 0 | 68 | CHEMBL3545131 |
| Porfimer | — | — | 10 | 0 | 25 | — |
| Vinblastine | Small Molecule | Tubulin inhibitor | 10 | 0 | 141 | CHEMBL159 |
| Vemurafenib | Small Molecule | Serine/threonine-protein kinase B-raf inhibitor | 9 | 261 | 119 | C64768 · CHEMBL1229517 |
| Neratinib | Small Molecule | Epidermal growth factor receptor erbB1 inhibitor; Receptor protein-tyrosine kinase erbB-2 inhibitor; Receptor protein-tyrosine kinase erbB-4 inhibitor | 9 | 43 | 71 | C49094 · CHEMBL180022 |
| Brigatinib | Small Molecule | ALK tyrosine kinase receptor inhibitor; Epidermal growth factor receptor erbB1 inhibitor | 9 | 21 | 34 | C98831 · CHEMBL3545311 |
| Ivosidenib | Small Molecule | Isocitrate dehydrogenase [NADP] cytoplasmic inhibitor | 9 | 16 | 46 | C114383 · CHEMBL3989958 |
| Daunorubicin | Small Molecule | DNA topoisomerase II alpha inhibitor; DNA inhibitor | 9 | 15 | 252 | C62091 · CHEMBL178 |
| Niraparib | Small Molecule | Poly [ADP-ribose] polymerase 2 inhibitor; Poly [ADP-ribose] polymerase-1 inhibitor | 9 | 13 | 173 | C80059 · CHEMBL1094636 |
| Avapritinib | Small Molecule | Stem cell growth factor receptor inhibitor; Platelet-derived growth factor receptor alpha inhibitor | 9 | 3 | 22 | C123827 · CHEMBL4204794 |
| Sorafenib Tosylate | Small Molecule | Serine/threonine-protein kinase RAF inhibitor; Platelet-derived growth factor receptor beta inhibitor; Stem cell growth factor receptor inhibitor; Tyrosine-protein kinase receptor FLT3 inhibitor; Serine/threonine-protein kinase B-raf inhibitor; Vascular endothelial growth factor receptor inhibitor; Tyrosine-protein kinase receptor RET inhibitor | 9 | 1 | 135 | C2194 · CHEMBL1200485 |
| Aminolevulinic Acid | Small Molecule | DNA inhibitor | 9 | 0 | 41 | CHEMBL601 |
| Cinacalcet | Small Molecule | Calcium sensing receptor positive allosteric modulator | 9 | 0 | 6 | CHEMBL1201284 |
| Entrectinib | Small Molecule | Neurotrophic tyrosine kinase receptor inhibitor; Proto-oncogene tyrosine-protein kinase ROS inhibitor; ALK tyrosine kinase receptor inhibitor | 8 | 73 | 33 | C114984 · CHEMBL1983268 |
| Erdafitinib | Small Molecule | Fibroblast growth factor receptor inhibitor | 8 | 56 | 26 | C103273 · CHEMBL3545376 |
| Binimetinib | Small Molecule | Dual specificity mitogen-activated protein kinase kinase 1 inhibitor; Dual specificity mitogen-activated protein kinase kinase 2 inhibitor | 8 | 24 | 100 | C84865 · CHEMBL3187723 |
| Trastuzumab Emtansine | Adc | Receptor protein-tyrosine kinase erbB-2 binding agent; Tubulin inhibitor | 8 | 19 | 126 | C82492 · CHEMBL1743082 |
| Abiraterone | Small Molecule | Cytochrome P450 17A1 inhibitor; Androgen Receptor antagonist; Steroid 5-alpha-reductase inhibitor | 8 | 14 | 111 | C77333 · CHEMBL254328 |