Loading drugs…
Loading drugs…
Drugs
One entity per molecule (INN preferred); brand names and development codes are aliases. Approvals are always shown with jurisdiction and indication.
819 drugs
| Drug | Kind | Mechanism | Approvals | Evidence items | Trials | Identifiers |
|---|---|---|---|---|---|---|
| Zanubrutinib | Small Molecule | Tyrosine-protein kinase BTK inhibitor | 23 | 0 | 121 | CHEMBL3936761 |
| Fluorouracil | Small Molecule | Thymidylate synthase inhibitor; DNA inhibitor; RNA inhibitor | 22 | 43 | 1,324 | C505 · CHEMBL185 |
| Tofacitinib | Small Molecule | Janus Kinase (JAK) inhibitor | 22 | 1 | 16 | C95800 · CHEMBL221959 |
| Interferon Beta-1a | Other | Interferon alpha/beta receptor agonist | 22 | 0 | 2 | CHEMBL1201562 |
| Trastuzumab Deruxtecan | Adc | Receptor protein-tyrosine kinase erbB-2 binding agent; DNA topoisomerase I inhibitor | 21 | 24 | 14 | C128799 · CHEMBL4297844 |
| Trastuzumab Deruxtecan | Adc | Receptor protein-tyrosine kinase erbB-2 binding agent; DNA topoisomerase I inhibitor | 21 | 3 | 0 | C152716 · CHEMBL4297844 |
| Lenalidomide | Small Molecule | CRL4(CRBN) E3 ubiquitin ligase inhibitor; CRL4(CRBN) E3 ubiquitin ligase modulator | 21 | 1 | 863 | C2668 · CHEMBL848 |
| Afatinib | Small Molecule | Epidermal growth factor receptor erbB1 inhibitor; Receptor protein-tyrosine kinase erbB-2 inhibitor; Receptor protein-tyrosine kinase erbB-4 inhibitor | 20 | 132 | 163 | C66940 · CHEMBL1173655 |
| Cabozantinib | Small Molecule | Vascular endothelial growth factor receptor 2 inhibitor; Hepatocyte growth factor receptor inhibitor | 20 | 19 | 246 | C52200 · CHEMBL2105717 |
| Ruxolitinib | Small Molecule | Tyrosine-protein kinase JAK1 inhibitor; Tyrosine-protein kinase JAK2 inhibitor; Tyrosine-protein kinase JAK3 inhibitor; Tyrosine-protein kinase TYK2 inhibitor | 20 | 14 | 177 | C77888 · CHEMBL1789941 |
| Daratumumab | Monoclonal Antibody | Lymphocyte differentiation antigen CD38 inhibitor | 19 | 0 | 261 | CHEMBL1743007 |
| Venetoclax | Small Molecule | Apoptosis regulator Bcl-2 inhibitor | 18 | 37 | 589 | C103147 · CHEMBL3137309 |
| Etoposide | Small Molecule | DNA topoisomerase II inhibitor | 18 | 10 | 1,197 | C491 · CHEMBL44657 |
| Arsenic Trioxide | Small Molecule | Thioredoxin reductase 1 inhibitor | 18 | 6 | 113 | C1005 · CHEMBL5483015 |
| Abemaciclib | Small Molecule | Cyclin-dependent kinase 4 inhibitor; Cyclin-dependent kinase 6 inhibitor | 18 | 5 | 195 | C97660 · CHEMBL3301610 |
| Cemiplimab | Monoclonal Antibody | Programmed cell death protein 1 inhibitor | 18 | 0 | 191 | CHEMBL4297723 |
| Crizotinib | Small Molecule | Hepatocyte growth factor receptor inhibitor; ALK tyrosine kinase receptor inhibitor; EML4-ALK inhibitor; NPM/ALK (Nucleophosmin/ALK tyrosine kinase receptor) inhibitor; Proto-oncogene tyrosine-protein kinase ROS inhibitor; Macrophage-stimulating protein receptor inhibitor | 17 | 267 | 100 | C74061 · CHEMBL601719 |
| Pertuzumab | Monoclonal Antibody | Receptor protein-tyrosine kinase erbB-2 inhibitor | 17 | 24 | 239 | C38692 · CHEMBL2007641 |
| Talazoparib | Small Molecule | Poly [ADP-ribose] polymerase 2 inhibitor; Poly [ADP-ribose] polymerase-1 inhibitor | 17 | 24 | 99 | C95733 · CHEMBL3137320 |
| Epirubicin | Small Molecule | DNA inhibitor | 17 | 1 | 285 | C62028 · CHEMBL417 |
| Nintedanib | Small Molecule | Platelet-derived growth factor receptor inhibitor; Vascular endothelial growth factor receptor inhibitor; Fibroblast growth factor receptor inhibitor | 17 | 1 | 71 | C62765 · CHEMBL502835 |
| Peginterferon Alfa-2b | Other | Interferon alpha/beta receptor agonist | 17 | 1 | 50 | C1845 · CHEMBL1201561 |
| Tislelizumab | Monoclonal Antibody | Programmed cell death protein 1 inhibitor | 17 | 1 | 407 | C152661 · CHEMBL4297840 |
| Thiotepa | Small Molecule | DNA inhibitor | 17 | 0 | 182 | CHEMBL671 |
| Cisplatin | Small Molecule | DNA inhibitor | 16 | 78 | 2,504 | C376 · CHEMBL11359 |
| Osimertinib | Small Molecule | Epidermal growth factor receptor erbB1 inhibitor | 16 | 62 | 223 | C116377 · CHEMBL3353410 |
| Sirolimus | Small Molecule | FK506-binding protein 1A inhibitor | 16 | 32 | 230 | C1212 · CHEMBL413 |
| Aflibercept | Other | Vascular endothelial growth factor A inhibitor; Placenta growth factor inhibitor | 16 | 0 | 75 | CHEMBL1742982 |
| Brentuximab Vedotin | Adc | Tubulin inhibitor; Tumor necrosis factor receptor superfamily member 8 binding agent | 16 | 0 | 167 | CHEMBL1742994 |
| Interferon Alfa-2b | Other | Interferon alpha/beta receptor agonist | 16 | 0 | 24 | CHEMBL1201558 |
| Cetuximab | Monoclonal Antibody | Epidermal growth factor receptor erbB1 inhibitor | 15 | 403 | 782 | C1723 · CHEMBL1201577 |
| Bosutinib | Small Molecule | Tyrosine-protein kinase ABL inhibitor; Tyrosine-protein kinase SRC inhibitor; Tyrosine-protein kinase HCK inhibitor; Tyrosine-protein kinase Lyn inhibitor; Bcr/Abl fusion protein inhibitor | 15 | 91 | 41 | C60809 · CHEMBL288441 |
| Encorafenib | Small Molecule | Serine/threonine-protein kinase B-raf inhibitor | 15 | 14 | 68 | C98283 · CHEMBL3301612 |
| Amivantamab | Monoclonal Antibody | Epidermal growth factor receptor erbB1 inhibitor; Hepatocyte growth factor receptor inhibitor | 15 | 5 | 40 | C124993 · CHEMBL4297774 |
| Acalabrutinib | Small Molecule | Tyrosine-protein kinase BTK inhibitor | 15 | 0 | 117 | CHEMBL3707348 |
| Tretinoin | Small Molecule | Retinoic acid receptor agonist | 14 | 14 | 102 | C900 · CHEMBL38 |
| Ramucirumab | Monoclonal Antibody | Vascular endothelial growth factor receptor 2 inhibitor | 14 | 3 | 137 | C70792 · CHEMBL1743062 |
| Carfilzomib | Other | 26S proteasome inhibitor | 14 | 1 | 208 | C52196 · CHEMBL451887 |
| Ibuprofen | Small Molecule | Cyclooxygenase inhibitor | 14 | 1 | 20 | C561 · CHEMBL521 |
| Peginterferon Alfa-2a | Other | Interferon alpha/beta receptor agonist | 14 | 1 | 18 | C33987 · CHEMBL1201560 |
| Zoledronic Acid | Small Molecule | Farnesyl diphosphate synthase inhibitor | 14 | 1 | 178 | C1699 · CHEMBL4303669 |
| Megestrol | Small Molecule | Progesterone receptor agonist | 14 | 0 | 43 | CHEMBL1201139 |
| Sorafenib | Small Molecule | Serine/threonine-protein kinase RAF inhibitor; Platelet-derived growth factor receptor beta inhibitor; Stem cell growth factor receptor inhibitor; Tyrosine-protein kinase receptor FLT3 inhibitor; Serine/threonine-protein kinase B-raf inhibitor; Vascular endothelial growth factor receptor inhibitor; Tyrosine-protein kinase receptor RET inhibitor | 13 | 96 | 443 | C61948 · CHEMBL1336 |
| Carboplatin | Small Molecule | DNA inhibitor | 13 | 38 | 2,385 | C1282 · CHEMBL1351 |
| Melphalan | Small Molecule | DNA inhibitor | 13 | 25 | 578 | C633 · CHEMBL852 |
| Cabazitaxel | Small Molecule | Tubulin inhibitor | 13 | 3 | 104 | C66937 · CHEMBL1201748 |
| Sacituzumab Govitecan | Adc | Tumor-associated calcium signal transducer 2 binding agent; DNA topoisomerase I inhibitor | 13 | 3 | 119 | C102783 · CHEMBL3545262 |
| Idarubicin | Small Molecule | DNA topoisomerase II alpha inhibitor; DNA inhibitor | 13 | 1 | 193 | C562 · CHEMBL1117 |
| Osimertinib Mesylate | Small Molecule | Epidermal growth factor receptor erbB1 inhibitor | 13 | 1 | 5 | C170266 · CHEMBL3545063 |
| Blinatumomab | Monoclonal Antibody | T cell surface glycoprotein CD3 cross-linking agent; B-lymphocyte antigen CD19 cross-linking agent | 13 | 0 | 141 | CHEMBL1742992 |