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Metabolic Activation-Dependent Anti-Liver Cancer Activity and Organ-Specific Toxicity of Retrorsine From Fanhuncao (Jacobaea cannabifolia and J. litvinovii).

Zhijie He, Zhongyu Tan, Lunrong Zhang, Yue Yin, Yedeli Yerjiang, Bo Bi, Jingshan Bao

Archiv der PharmazieSep 1, 2026PMID 42704289doi:10.1002/ardp.70326 PMC13548937Journal ArticlepubmedProvenance
Source
PubMed
Retrieved
Sep 14, 2026
Layer
normalized (units and labels harmonized; values unchanged)
Run
ING-PUBMED-20260914-000001
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Fanhuncao (Jacobaea cannabifolia and J. litvinovii) is a traditional Chinese herb with reported antitumor potential. Retrorsine, a pyrrolizidine alkaloid from Fanhuncao, requires CYP3A4‑mediated metabolic activation, but its dual outcomes (anti‑liver cancer efficacy vs. organ‑specific toxicity)…

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