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Drugs
One entity per molecule (INN preferred); brand names and development codes are aliases. Approvals are always shown with jurisdiction and indication.
820 drugs
| Drug | Kind | Mechanism | Approvals | Evidence items | Trials | Identifiers |
|---|---|---|---|---|---|---|
| EFTX-G12V | — | — | 0 | 1 | 0 | — |
| EGFR Tyrosine Kinase Inhibitor Therapy | — | — | 0 | 1 | 0 | C116534 |
| Endocrine Drug Therapy | — | — | 0 | 1 | 0 | C63475 |
| Enzastaurin | Small Molecule | Protein kinase C beta inhibitor | 0 | 1 | 48 | C77392 · CHEMBL300138 |
| EPZ004777 | Small Molecule | — | 0 | 1 | 0 | CHEMBL2169919 |
| ERBB3 Inhibitor | — | — | 0 | 1 | 0 | — |
| Erdafitinib Regimen | — | — | 0 | 1 | 0 | C186501 |
| EZH2 Inhibitor | Small Molecule | — | 0 | 1 | 0 | C156804 · CHEMBL3414574 |
| FAC Regimen | — | — | 0 | 1 | 1 | C138099 |
| FACT Complex-targeting Curaxin CBL0137 | — | — | 0 | 1 | 5 | C107239 |
| Fadraciclib | Small Molecule | — | 0 | 1 | 6 | C123902 · CHEMBL3655762 |
| Fasudil | Small Molecule | Rho-associated protein kinase inhibitor | 0 | 1 | 2 | C65624 · CHEMBL38380 |
| FEC Regimen | — | — | 0 | 1 | 0 | C63420 |
| FGFR4 Inhibitor H3B-6527 | — | — | 0 | 1 | 1 | C128862 |
| FGFR Inhibitor ASP5878 | — | — | 0 | 1 | 1 | C122719 |
| Fisogatinib | Small Molecule | — | 0 | 1 | 1 | C123826 · CHEMBL4514636 |
| FOLFIRI-Panitumumab Regimen | — | — | 0 | 1 | 0 | C136249 |
| FOLFOX-6 Regimen | — | — | 0 | 1 | 9 | C63591 |
| FOLFOX Regimen | — | — | 0 | 1 | 163 | C11197 |
| G007-LK | — | — | 0 | 1 | 0 | — |
| G-573 | — | — | 0 | 1 | 0 | — |
| Galeterone | Small Molecule | Androgen Receptor antagonist; Cytochrome P450 17A1 inhibitor | 0 | 1 | 4 | C84866 · CHEMBL2105738 |
| Galiximab | Monoclonal Antibody | T-lymphocyte activation antigen CD80 inhibitor | 0 | 1 | 5 | C26447 · CHEMBL2109191 |
| GDC-0879 | Small Molecule | — | 0 | 1 | 0 | CHEMBL525191 |
| GF109203X | — | — | 0 | 1 | 0 | — |
| GNE-617 | Small Molecule | — | 0 | 1 | 0 | CHEMBL2420629 |
| Go6983 | — | — | 0 | 1 | 0 | — |
| GPI-15427 | — | — | 0 | 1 | 0 | — |
| G-Quadruplex Stabilizer BMVC | — | — | 0 | 1 | 0 | C95893 |
| GSK321 | — | — | 0 | 1 | 0 | — |
| Guadecitabine | Small Molecule | — | 0 | 1 | 27 | C95209 · CHEMBL3544916 |
| GW-2580 | — | — | 0 | 1 | 0 | — |
| HCI-2509 | — | — | 0 | 1 | 0 | — |
| HDAC Inhibitor OBP-801 | — | — | 0 | 1 | 1 | C121665 |
| HDM2 Inhibitor MK-8242 | — | — | 0 | 1 | 2 | C116867 |
| HER2 Inhibitor CP-724,714 | — | — | 0 | 1 | 2 | C26648 |
| HyperCVAD Regimen | — | — | 0 | 1 | 5 | C63455 |
| Hyperthermic Intraperitoneal Chemotherapy | — | — | 0 | 1 | 21 | C91835 |
| I-BET151 | Small Molecule | — | 0 | 1 | 0 | CHEMBL2017291 |
| ICX-101 | — | — | 0 | 1 | 0 | — |
| IMG-2005-5 | — | — | 0 | 1 | 0 | — |
| Immunomodulatory Oligonucleotide | — | — | 0 | 1 | 37 | — |
| Iniparib | Small Molecule | Reactive nitro radical | 0 | 1 | 13 | C62526 · CHEMBL1170047 |
| Interventional Radiology Procedure | — | — | 0 | 1 | 0 | C63334 |
| Iodine I-131 | — | — | 0 | 1 | 0 | C1639 |
| Ionizing Radiotherapy | — | — | 0 | 1 | 0 | C15846 |
| IRAK-1/4 Inhibitor | — | — | 0 | 1 | 0 | — |
| JAK2 Inhibitor AZD1480 | — | — | 0 | 1 | 2 | C91394 |
| JAK Inhibitor I | — | — | 0 | 1 | 0 | — |
| JNJ38877605 | — | — | 0 | 1 | 0 | — |